Abstract

A method for preparing 2-fluoro-3-aminobenzoic acid and an ester compound thereof. The reaction formula is as follows. Specifically, a compound I is nitrated under suitable reaction conditions to obtain a compound II; the compound II is halogenated under suitable reaction conditions to obtain a compound III; the compound III is fluorinated under suitable reaction conditions to obtain a compound IV; the compound IV is hydrolyzed or alcoholyzed under suitable reaction conditions to prepare a compound V; and the compound V is subjected to catalytic hydrogenation dehalogenation under suitable reaction conditions to obtain 2-fluoro-3-aminobenzoic acid and an ester compound thereof, namely a compound X. The starting material of the process route is cheap and easy to obtain, the procedures of the process are operated by common units in fine chemical industry, the operation is convenient, the reaction conversion rate is high, and the selectivity is good. The method provides an effective preparation method for industrial development of the compound.

IPC Classes  ?

• C07C 227/04 - Formation of amino groups in compounds containing carboxyl groups
• C07C 229/60 - Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring with amino and carboxyl groups bound in meta- or para- positions

Abstract

A preparation method for 2-fluoro-3-aminobenzoic acid and ester compounds thereof. A compound I is used as a raw material for nitration reaction to obtain a compound II; halogenation reaction is performed on the obtained compound II to obtain a compound III; fluorination is performed on the compound III under proper reaction conditions to obtain a compound IV; the obtained compound IV is prepared into a compound V in a hydrolysis or alcoholysis mode; catalytic hydrogenation dehalogenation is performed on the compound V to obtain 2-fluoro-3-aminobenzoic acid and ester compounds as shown in a compound X. According to the preparation method, the starting raw materials of the process route are cheap and easy to obtain, the technological process relates to common unit operation in fine chemical engineering, the operation is convenient, the reaction conversion rate is high, and the selectivity is good.

IPC Classes  ?

• C07C 227/04 - Formation of amino groups in compounds containing carboxyl groups
• C07C 229/60 - Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring with amino and carboxyl groups bound in meta- or para- positions

Abstract

Disclosed in the present invention are aryloxyphenoxypropionate compounds and the use thereof, the compounds being shown as general formula (I), and selection of substituents being described in detail in the specification. The compounds of the present invention not only have excellent herbicidal activity, but also are safe to crops.

IPC Classes  ?

• C07D 263/58 - BenzoxazolesHydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
• C07D 413/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 417/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/76 - 1,3-OxazolesHydrogenated 1,3-oxazoles

Abstract

The present invention relates to a herbicide composition and a use method therefor. The composition comprises two active ingredients A and B, wherein the weight ratio of the ingredient A to the ingredient B is 1:90-90:1; the ingredient A is selected from a compound represented by the following general formula. Stem and leaf spray treatments with the herbicide of the present invention can be used for the control of most weeds in places such as cultivated lands, uncultivated lands, orchards, idle cultivated lands, rubber plantations, eucalyptus forests, forests, firebreaks, lawns, railways, highways, airports, and warehouses.

IPC Classes  ?

• C07D 251/38 - Sulfur atoms
• A01N 43/66 - 1,3,5-Triazines, not hydrogenated and not substituted at the ring nitrogen atoms
• A01P 13/00 - HerbicidesAlgicides

Abstract

Disclosed are a synergistic insecticide composition containing a piperic acid derivative compound, and an application thereof. The composition is composed of two active ingredients, namely a compound A and a compound B, wherein the active ingredient A is compound I-72; and the active ingredient B is selected from one or more of: a nereistoxin insecticide, a macrolide insecticide, an organophosphorus insecticide, a carbamate insecticide, a quaternary keto acid insecticide, a nematicide, a biologically derived insecticide, a pyrethroid insecticide, a plant growth regulator, an insect attractant, a repellent, an insect growth regulator-type insecticide, an amide insecticide, a nicotine insecticide, an insect ingestion-blocking insecticide, a bactericide, an acaricide, or other insecticides and inorganic matter. The compound I-72 has the following structure: The composition of the present invention has advantages such as clear synergistic effect, delayed resistance, etc., and can be used for preventing and treating a variety of pests related to agriculture, forestry, and ornamental plants.

IPC Classes  ?

• A01N 43/30 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with two or more hetero atoms five-membered rings with two hetero atoms in positions 1,3 with two oxygen atoms in positions 1,3, condensed with a carbocyclic ring
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides

Abstract

The present invention belongs to the field of insecticides and acaricides, and relates to an insecticidal and acaricidal agent and the use thereof. The agent is a liquid agent, and contains at least one carrier and at least one auxiliary agent; and the agent is in a dosage form of an emulsion in water, a microemulsion, an emulsifiable concentrate and a soluble liquid or is an ultra-low volume agent, with a compound of formula I as an active component, wherein the active component of the insecticidal and acaricidal agent is the compound of formula I, the weight percentage content thereof being 0.1-90%. The active component compound A is a compound as shown in the following structural formula I.

IPC Classes  ?

• A01N 43/30 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with two or more hetero atoms five-membered rings with two hetero atoms in positions 1,3 with two oxygen atoms in positions 1,3, condensed with a carbocyclic ring
• A01N 25/22 - Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of applicationSubstances for reducing the noxious effect of the active ingredients to organisms other than pests containing ingredients stabilising the active ingredients
• A01N 25/02 - Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of applicationSubstances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides

Abstract

The present invention belongs to the technical field of agricultural insecticides, and relates to an insecticidal preparation containing a meta-diamide compound (as shown in general formula I) and the use thereof. The preparation contains an active ingredient, and contains at least one carrier and at least one auxiliary agent, characterized in that: the preparation is a suspension agent, a dispersible oil suspension agent, a dispersible liquid agent, a wettable powder, a water dispersible granule, or a dry suspension agent, wherein the active ingredient in the preparation is a compound as shown in general formula I, and accounts for 1%-99% by weight of the preparation. The insecticidal composition of the present invention has the characteristics of good wetting, spreading and penetration of the liquid pesticide on a target, less rebound of the liquid pesticide on a target, a large liquid holding amount, a large deposition amount, less evaporation, a large absorption rate, high biological activity, being safe for crops, etc., and is an ideal insecticide variety for preventing and controlling lepidoptera, coleoptera and thysanoptera and other pests.

IPC Classes  ?

• A01N 43/30 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with two or more hetero atoms five-membered rings with two hetero atoms in positions 1,3 with two oxygen atoms in positions 1,3, condensed with a carbocyclic ring
• C07D 317/46 - Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Abstract

The present invention pertains to the technical field of agricultural bactericides and particularly relates to a quinolinecarboxylic acid derivative and use thereof. The quinolinecarboxylic acid derivative is represented by general formula (I). The compound of general formula (I) shows good activity against various fungal diseases and bacterial diseases in the field of agriculture and can be used as a bactericide in the field of agriculture.

IPC Classes  ?

• C07D 215/56 - Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
• A01N 43/42 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
• A01P 1/00 - DisinfectantsAntimicrobial compounds or mixtures thereof

Abstract

Provided are a pyridazinone derivative and use thereof. The pyridazinone derivative is represented by general formula (I). The compound of general formula (I) has activity on various fungal diseases and bacterial diseases in the agricultural field, and can be used as a fungicide/bactericide in the agricultural field.

IPC Classes  ?

• C07D 237/18 - Sulfur atoms
• A01N 43/58 - 1,2-DiazinesHydrogenated 1,2-diazines
• A01P 3/00 - Fungicides

Abstract

The present invention belongs to the field of agricultural fungicides and bactericide, and specifically relates to an N-substituted aniline compound, and the uses thereof as a bactericide and a fungicide. The N-substituted aniline compound is represented by general formula (I), and the definition of each substituent in the formula is shown in the specification. The compound represented by general formula (I) shows good activity on various bacteria in the agricultural field, and particularly has excellent activity on diseases such as napa cabbage soft rot, muskmelon bacterial fruit blotch, cucumber bacterial angular leaf spot, tomato bacterial wilt, citrus canker, kiwi fruit canker, grape root cancer, rice bacterial leaf stripe, and tomato canker. In addition, the compound has low raw material cost, high cost performance and wide application prospect.

IPC Classes  ?

• A01N 33/18 - Nitro compounds
• C07C 211/56 - Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to two or three six-membered aromatic rings the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
• A01P 3/00 - Fungicides

Abstract

In a synthesis method of a phenylisoxazoline compound 2-fluoro-4-chloro-5-methylaniline is used as starting material for firstly synthesizing a uracil ring, and then synthesizing an isooxazoline ring to obtain a target compound, phenylisoxazoline compound (VII), as shown in the reaction pathway below. In a synthesis method of a phenylisoxazoline compound 2-fluoro-4-chloro-5-methylaniline is used as starting material for firstly synthesizing a uracil ring, and then synthesizing an isooxazoline ring to obtain a target compound, phenylisoxazoline compound (VII), as shown in the reaction pathway below. In a synthesis method of a phenylisoxazoline compound 2-fluoro-4-chloro-5-methylaniline is used as starting material for firstly synthesizing a uracil ring, and then synthesizing an isooxazoline ring to obtain a target compound, phenylisoxazoline compound (VII), as shown in the reaction pathway below. The preparation method can be used for the synthesis of phenylisoxazoline containing uracil.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 239/54 - Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals

Abstract

The present invention relates to a stabilizer-containing fungicidal composition preparation. The composition can be prepared into products of various dosage forms in combination with necessary formula components. After the product is subjected to an accelerated thermal storage test (54℃, 14d), the automatic dispersity of the sample in high-concentration hard water (hardness: 1000 ppm) can be improved (the automatic dispersity is higher than 95%), and the dilution stability and effective suspension rate under a low dilution ratio (20-time dilution) and high-hardness hard water conditions are increased (the effective suspension rate is higher than 95%).

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01N 25/22 - Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of applicationSubstances for reducing the noxious effect of the active ingredients to organisms other than pests containing ingredients stabilising the active ingredients

Abstract

The present invention belongs to the field of agricultural acaricides, and particularly relates to a substituted phenyl sulfide compound and an application thereof. The substituted phenyl sulfide compound is as represented in general formula I. Definitions of substituted groups in the formula are given in the description. The compound of the general formula I has excellent acaricidal activity and can be used for preventing and controlling various mites. The present invention belongs to the field of agricultural acaricides, and particularly relates to a substituted phenyl sulfide compound and an application thereof. The substituted phenyl sulfide compound is as represented in general formula I. Definitions of substituted groups in the formula are given in the description. The compound of the general formula I has excellent acaricidal activity and can be used for preventing and controlling various mites.

IPC Classes  ?

• C07C 317/32 - SulfonesSulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
• C07C 323/65 - Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and sulfur atoms, not being part of thio groups, bound to the same carbon skeleton containing sulfur atoms of sulfone or sulfoxide groups bound to the carbon skeleton
• A01P 7/02 - Acaricides

Abstract

A method for preparing an intermediate of a uracil compound containing isooxazoline includes the steps of: making 3-amino-4,4,4-trifluorocrotonic acid methyl ester react with substituted aryl carbamate; in a reaction process, continuously evaporating water and byproduct alcohol in the system; and conducting processing to obtain the intermediate of the uracil compound containing isooxazoline. Using this method the selectivity of the reaction and the utilization rate of raw materials are improved; the hydrolysis products, impurities and tar are reduced; the reaction time is greatly shortened; and the productivity is improved. After one recrystallization of crude products, an intermediate product with purity of more than 97% can be obtained, and quantitative yield can be more than 85%.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• B01J 31/02 - Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides

Abstract

The present invention discloses a triazine benzoate compound having the structure shown in formula (I) or a stereoisomer: The present invention discloses a triazine benzoate compound having the structure shown in formula (I) or a stereoisomer: The present invention discloses a triazine benzoate compound having the structure shown in formula (I) or a stereoisomer: The definition of each substituent in the formula I is described in the description. The compound of the formula I of the present invention has excellent herbicidal activity and can be used for controlling weeds.

IPC Classes  ?

• C07D 251/32 - Cyanuric acidIsocyanuric acid
• C07D 251/38 - Sulfur atoms
• C07D 405/12 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01P 13/00 - HerbicidesAlgicides
• A01N 43/64 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms

Abstract

The present invention discloses an amide compound containing substituted acetophenone structural fragments, having a structure shown by general formula I: The present invention discloses an amide compound containing substituted acetophenone structural fragments, having a structure shown by general formula I: The present invention discloses an amide compound containing substituted acetophenone structural fragments, having a structure shown by general formula I: The definitions of substituents in the formula are shown in the description. The compound of the present invention has broad-spectrum fungal activity, and has excellent control effects on cucumber downy mildew, wheat powdery mildew, corn rust, cucumber anthracnose, cucumber botrytis and tomato botrytis.

IPC Classes  ?

• C07D 213/82 - AmidesImides in position 3
• C07D 231/12 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
• C07D 231/16 - Halogen atoms or nitro radicals

Abstract

An alkene-containing carboxylic ester compound of formula (I) and its agriculturally acceptable salt can be used as a herbicide. An alkene-containing carboxylic ester compound of formula (I) and its agriculturally acceptable salt can be used as a herbicide.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 231/20 - One oxygen atom attached in position 3 or 5
• C07D 405/12 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 231/24 - One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms having sulfone or sulfonic acid radicals in the molecule
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 403/10 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 401/10 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 401/06 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
• C07D 405/14 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
• C07D 413/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 47/06 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom containing —O—CO—O— groupsThio-analogues thereof
• A01N 47/12 - Carbamic acid derivatives, i.e. containing the group —O—CO—NThio-analogues thereof containing a —O—CO—N group, or a thio-analogue thereof, neither directly attached to a ring nor the nitrogen atom being a member of a heterocyclic ring
• A01N 47/30 - Derivatives containing the group N—CO—N—aryl or N—CS—N—aryl
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

Pyrazole carboxylate ester compounds have a structural formula of formula (I): Pyrazole carboxylate ester compounds have a structural formula of formula (I): Pyrazole carboxylate ester compounds have a structural formula of formula (I): Q is Q1 or Q3 Pyrazole carboxylate ester compounds have a structural formula of formula (I): Q is Q1 or Q3 Pyrazole carboxylate ester compounds have a structural formula of formula (I): Q is Q1 or Q3 The pyrazole carboxylate ester compounds has herbicidal activity and can be used for controlling weeds.

IPC Classes  ?

• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention belongs to the field of insecticides and acaricides, and specifically relates to an imine compound and the use thereof. The structure is as represented by general formula I, wherein each substituent in the formula is defined in the description. The compound of general formula I has excellent insecticidal and acaricidal activities, and can be used for preventing and controlling various pest insects or pest mites.

IPC Classes  ?

• C07C 257/02 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by halogen atoms, e.g. imino-halides
• C07C 257/00 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
• C07C 257/10 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
• C07C 237/40 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having the nitrogen atom of the carboxamide group bound to a carbon atom of a six-membered aromatic ring
• C07C 235/56 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
• C07D 317/46 - Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
• A01N 37/22 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N, e.g. carboxylic acid amides or imidesThio-analogues thereof the nitrogen atom being directly attached to an aromatic ring system, e.g. anilides
• A01N 37/38 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio-analogue, or a derivative thereof, and a singly bound oxygen or sulfur atom attached to the same carbon skeleton, this oxygen or sulfur atom not being a member of a carboxylic group or of a thio-analogue, or of a derivative thereof, e.g. hydroxy-carboxylic acids having at least one oxygen or sulfur atom attached to an aromatic ring system
• A01P 7/02 - Acaricides

Abstract

An alkene-containing amide compound of formula (I) and agriculturally acceptable salts thereof can be used as herbicides. An alkene-containing amide compound of formula (I) and agriculturally acceptable salts thereof can be used as herbicides.

IPC Classes  ?

• C07D 257/06 - Five-membered rings with nitrogen atoms directly attached to the ring carbon atom
• A01N 43/713 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
• C07D 405/12 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 413/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 43/82 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with three hetero atoms
• C07D 271/113 - 1,3,4-OxadiazolesHydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
• C07D 285/135 - Nitrogen atoms
• C07D 249/14 - Nitrogen atoms
• C07D 271/04 - 1,2,3-OxadiazolesHydrogenated 1,2,3-oxadiazoles
• C07D 413/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• C07D 417/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention belongs to the field of agricultural herbicides, and relates to a dispersible oil suspension of a herbicide composition and a preparation method therefor. The present invention also relates to a use of the dispersible oil suspension for preventing unwanted plant growth. The dispersible oil suspension has the following components according to weight percentage: 0.1% to 20% of active component A, 1% to 60% of active component B, 1% to 30% of a surfactant, 0.1 to 5% of a pH adjuster, 0.5% to 5% of a structurally stable agent, 0 to 20% of a solvent, and the remainder is an oil base. The active component A is a compound shown in formula I, and the active component B is selected from glyphosate and salts or esters agrochemically applicable thereto. The dispersible oil suspension provided by the present invention is stable, has no physical instability phenomena such as livering and bottoming during thermal storage, and the effective components do not easily decompose. The herbicide composition of the present invention may be used to control various weeds, especially broadleaf weeds, such as abutilon and common zinnia, and has excellent control effects.

IPC Classes  ?

• A01N 57/20 - Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-carbon bonds containing acyclic or cycloaliphatic radicals
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 25/04 - Dispersions or gels
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention discloses an oxime ether compound with novel structure. The structure is shown in general formula I. The definition of each substituent in the formula is provided in the description. The present invention discloses an oxime ether compound with novel structure. The structure is shown in general formula I. The definition of each substituent in the formula is provided in the description. The present invention discloses an oxime ether compound with novel structure. The structure is shown in general formula I. The definition of each substituent in the formula is provided in the description. The compound of general formula I has excellent microbicidal 1 activity, and has good control effects on plant bacterial diseases and fungal diseases. The present invention comprises an application of the compound of the general formula I as a microbicide in agriculture and other fields.

IPC Classes  ?

• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• C07D 277/46 - Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
• C07D 277/40 - Unsubstituted amino or imino radicals
• C07D 277/50 - Nitrogen atoms bound to hetero atoms
• A01P 1/00 - DisinfectantsAntimicrobial compounds or mixtures thereof
• A01P 3/00 - Fungicides

Abstract

An isoxazoline compound with optical activity is shown in the formula (I). The compound of the formula (I) has excellent herbicidal activity, can be used for weeding pre- and post-emergence, and can also be used for soil treatment. The compound of the formula (I) can effectively control various broad-leaved weeds, grass weeds and Cyperaceae weeds, and can control various resistant weeds, such as glyphosate-resistant weeds. The excellent weeding effect can be obtained at a low dose. The compound has good safety to crops such as corn, wheat, rice, soybean and sugar beet. The compound can be used as a selective herbicide in crop fields in agriculture, and can also be used as a non-selective herbicide in non-cultivated land, fallow land, woodland, orchards and ridges. An isoxazoline compound with optical activity is shown in the formula (I). The compound of the formula (I) has excellent herbicidal activity, can be used for weeding pre- and post-emergence, and can also be used for soil treatment. The compound of the formula (I) can effectively control various broad-leaved weeds, grass weeds and Cyperaceae weeds, and can control various resistant weeds, such as glyphosate-resistant weeds. The excellent weeding effect can be obtained at a low dose. The compound has good safety to crops such as corn, wheat, rice, soybean and sugar beet. The compound can be used as a selective herbicide in crop fields in agriculture, and can also be used as a non-selective herbicide in non-cultivated land, fallow land, woodland, orchards and ridges.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2

Abstract

The present invention belongs to the field of agricultural herbicides, and particularly relates to an aryl isoxazoline compound and a use thereof. The aryl isoxazoline compound is represented by general formula (I). The compound of general formula (I) has good herbicidal activity, can effectively control gramineae and broadleaf weeds, can achieve good weeding effects at a low dose, is safe for crops such as corn, wheat, soybean and the like, and can be used as a herbicide in agriculture.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 413/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention belongs to the fields of insecticides and acaricides, and particularly relates to a piperonylic acid derivative and application thereof. The structure is shown in a general formula I, and the definition of each substituent in the formula is described in the description. The compound of the general formula I has excellent insecticidal and acaricidal activity and can be used for controlling various pests and mites. The present invention belongs to the fields of insecticides and acaricides, and particularly relates to a piperonylic acid derivative and application thereof. The structure is shown in a general formula I, and the definition of each substituent in the formula is described in the description. The compound of the general formula I has excellent insecticidal and acaricidal activity and can be used for controlling various pests and mites.

IPC Classes  ?

• A01N 43/30 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with two or more hetero atoms five-membered rings with two hetero atoms in positions 1,3 with two oxygen atoms in positions 1,3, condensed with a carbocyclic ring
• C07D 317/46 - Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
• A01P 7/04 - Insecticides

Abstract

The present invention relates to a herbicide composition and the use method thereof, wherein component A is a compound as represented by structural formula I. Component B is selected from one or more of ALS inhibitors, ACCa enzyme inhibitors, HPPD inhibitors, triazinones, PPO inhibitors, and hormone inhibitor herbicides. The herbicide composition of the present invention is applied to a locus where unwanted vegetation is present or expected to be present; and same is particularly suitable for the prevention and elimination of non-cultivated weeds.

IPC Classes  ?

• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01N 41/10 - SulfonesSulfoxides
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 47/30 - Derivatives containing the group N—CO—N—aryl or N—CS—N—aryl
• A01N 47/36 - Ureas or thioureas containing the groups N—CO—N or N—CS—N containing the group N—CO—N directly attached to at least one heterocyclic ringThio-analogues thereof
• A01N 47/38 - Ureas or thioureas containing the groups N—CO—N or N—CS—N containing the group N—CO—N where at least one nitrogen atom is part of a heterocyclic ringThio-analogues thereof
• A01N 43/90 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
• A01N 43/64 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
• A01N 41/06 - Sulfonic acid amides
• A01N 43/707 - 1,2,3- or 1,2,4-TriazinesHydrogenated 1,2,3- or 1,2,4-triazines
• A01N 33/22 - Nitro compounds containing oxygen or sulfur attached to the carbon skeleton containing the nitro group having at least one oxygen or sulfur atom and at least one nitro group directly attached to the same aromatic ring system
• A01P 13/00 - HerbicidesAlgicides

Abstract

Provided are a method of preparing a malononitrile oxime ether compound and an intermediate compound. The malononitrile oxime ether compound has a structure as shown in formula (VII), wherein W is selected from aryl or heteroaryl. The preparation method comprises: reacting a first raw material with a second raw material in the presence of a first solvent and a catalyst to obtain the intermediate compound, wherein the first raw material has a structure as shown in formula (IV), and the second raw material has a structure as shown in formula (V); and subjecting the intermediate compound, and a dehydrant to a dehydration reaction in the present of a second solvent to obtain the malononitrile oxime ether compound. Furthermore, the malononitrile oxime ether compound is obtained through one-step dehydration reaction. using the preparation method, is advantageous for improving the yield of malononitrile oxime ethers and reducing the cost.

IPC Classes  ?

• C07D 277/24 - Radicals substituted by oxygen atoms
• C07C 253/20 - Preparation of carboxylic acid nitriles by dehydratation of carboxylic acid amides
• C07C 253/30 - Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
• C07C 255/64 - Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton with the nitrogen atoms further bound to oxygen atoms
• C07D 213/61 - Halogen atoms or nitro radicals
• C07D 215/14 - Radicals substituted by oxygen atoms

Abstract

A preparation method for a bromopyrazole carboxylate compound. The chemical formula is as shows below, formula (I), formula (II), and the definition of each group in the formula is shown in the specification. A method for preparing a bromopyrazole carboxylate compound as a key intermediate in benzamide insecticides. The method is simple and easy to operate, safer, more reliable, and easier for industrial production.

IPC Classes  ?

• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond
• C07D 231/06 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
• C07D 231/08 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with oxygen or sulfur atoms directly attached to ring carbon atoms

Abstract

The present invention belongs to the field of organic synthesis, and particularly relates to a method for preparing a mesotrione herbicide. 4-methanesulfonyl-2-nitrobenzoic acid is used as a raw material, and is subjected to a chloroformylation reaction and an esterification reaction to obtain a reaction system containing an enol ester, followed by a rearrangement reaction to prepare mesotrione, that is, a rearrangement catalyst is added into the reaction system containing the enol ester, same is maintained at 0-40ºC and subjected to the rearrangement reaction, so as to obtain mesotrione. According to the method of the present invention, the use of a highly toxic acetone cyanohydrin rearrangement catalyst is avoided, the reaction temperature is appropriate, the reaction time is short, the solvent can be recycled, the total yield of the prepared mesotrione herbicide product can reach 89%, the content is 98%, and the process is safe and environmentally-friendly, creates a small amount of the three wastes, and is suitable for industrial production.

IPC Classes  ?

• C07C 315/04 - Preparation of sulfonesPreparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
• C07C 317/24 - SulfonesSulfoxides having sulfone or sulfoxide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
• C07C 317/44 - SulfonesSulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton

Abstract

The present invention relates to the field of agricultural acaricides, and in particular to a substituted phenyl sulfide compound and an application thereof. The substituted phenyl sulfide compound is as represented by general formula I. Definitions of substituted groups in the formula are given in the description. The compound of general formula I has excellent acaricidal activities and can be used for preventing and controlling various mites.

IPC Classes  ?

• C07C 317/14 - SulfonesSulfoxides having sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings
• C07C 309/00 - Sulfonic acidsHalides, esters, or anhydrides thereof
• C07C 317/32 - SulfonesSulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
• C07C 323/31 - Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
• C07C 323/09 - Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
• C07C 317/22 - SulfonesSulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
• A01P 7/02 - Acaricides

Abstract

The present invention belongs to the field of organic synthesis. The present invention provides a synthesis method of a phenylisoxazoline compound. 2-fluoro-4-chloro-5-methylaniline is used as starting material for firstly synthesizing a uracil ring, and then synthesizing an isooxazoline ring to obtain a target compound, phenylisoxazoline compound (VII). The definition of each group in the formula is explained in the description. The preparation method provided by the present invention can be widely used for the synthesis of phenylisoxazoline containing uracil, greatly improves the yield, effectively reduces the cost, and is easy to industrial production.

IPC Classes  ?

• C07D 239/54 - Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

The present invention relates to a preparation method of a class of herbicide intermediates, in particular to a method for preparing an intermediate of a uracil compound containing isooxazoline, which comprises: making 3-amino-4,4,4-trifluorocrotonic acid methyl ester react with substituted aryl carbamate; in a reaction process, continuously evaporating water and byproduct alcohol in the system; and conducting processing to obtain the intermediate of the uracil compound containing isooxazoline. In the method of the present invention, the selectivity of the reaction and the utilization rate of raw materials are improved; the hydrolysis products, impurities and tar are reduced; the reaction time is greatly shortened; and the productivity is improved. Moreover, after one recrystallization of crude products, an intermediate product with purity of more than 97% can be obtained, and quantitative yield can be more than 85%, which is suitable for industrial production.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

The present invention provides a synthesis method for a phenylisoxazoline compound, comprising: synthesizing uracil first by taking 2-fluoro-4-chloro-5-methylaniline as a starting raw material, and then synthesizing an isoxazoline ring to obtain a target compound, i.e., the phenylisoxazoline compound. The preparation method provided in the present invention can be widely used for synthesizing phenylisoxazoline containing uracil, and can greatly improve the yield, effectively reduce the cost, and facilitate industrial production.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 239/54 - Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals

Abstract

The present invention relates to a method for preparing a class of herbicide intermediates, specifically a method for preparing isoxazoline-containing uracil compound intermediates: reacting 3-amino-4, 4, 4-trifluorocrotonate and substituted aryl carbamate, the reaction process continuously steaming off water and by-product alcohol in the system and, after treament, obtaining an isoxazoline-containing uracil compound intermediate. The method of the present invention greatly increases the selectivity of the reaction and the rate of utilisation of the raw materials, reduces the hydrolysate and the production of impurities and tar, greatly shortens the reaction time and increases productivity, can obtain an intermediate product with purity of more than 97% by subjecting the crude product to one recrystallisation, can reach a quantitative yield of more than 86%, and is suitable for industrial production.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

Disclosed in the present invention is a triazine benzoate compound, having a structure as shown in general formula (I) or a stereoisomer thereof. The definition of substituents in general formula I is described in the description. The compound of general formula I of the present invention has excellent herbicidal activity and can be used for preventing and treating weeds.

IPC Classes  ?

• C07D 251/38 - Sulfur atoms
• A01N 43/66 - 1,3,5-Triazines, not hydrogenated and not substituted at the ring nitrogen atoms
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention discloses a triazine benzoate compound having the structure shown in formula (I) or a stereoisomer: (I) The definition of each substituent in the formula I is described in the description. The compound of the formula I of the present invention has excellent herbicidal activity and can be used for controlling weeds.

IPC Classes  ?

• A01N 43/66 - 1,3,5-Triazines, not hydrogenated and not substituted at the ring nitrogen atoms
• C07D 251/38 - Sulfur atoms

Abstract

133. See the description for the definition of each substituent in general formula (I). The compound of general formula I of the present invention has a good herbicidal activity and can be used for the control of weeds.

IPC Classes  ?

• C07D 231/14 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 231/16 - Halogen atoms or nitro radicals
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles

Abstract

Disclosed are a pyrazole carboxylate compound and the use thereof. The compound is as shown by general formula (I): wherein Q is the following groups: Q1 or Q3. See the description for the definition of each substituent in general formula (I). The compound of general formula I of the present invention has a good herbicidal activity and can be used for the control of weeds.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 231/14 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 231/16 - Halogen atoms or nitro radicals

Abstract

Provided is a one-step method for preparing imidazolinone compound (I), comprising putting a quaternary ammonium salt compound of general formula II and 2-amino-2,3-dimethylbutanamide in a suitable solvent to perform a reaction in the presence of a base at a temperature within the range of 0°C to the boiling point of the suitable solvent, and after the reaction, obtaining the imidazolinone compound (I) by means of acidification. According to the method, the reaction steps is refuced, the operation process is simplified, the reaction conditions are mild, the volume of the three wastes (waste gas, waste water, and industrial residue) is reduced, and the product content is high.

IPC Classes  ?

• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond
• A01N 47/36 - Ureas or thioureas containing the groups N—CO—N or N—CS—N containing the group N—CO—N directly attached to at least one heterocyclic ringThio-analogues thereof
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention falls within the field of agricultural bactericides. Specifically disclosed are a bactericidal composition and the use thereof. The composition is composed of two active components: A and B. The weight ratio between active component A and active component B is 1:99-99:1; and active component A is one or more of pyrimidine-containing substituted pyrazole compounds or salts thereof, and active component B is selected from a bactericide. The bactericidal composition of the present invention is particularly suitable for preventing and controlling various plant pathogenic fungi and bacterial diseases.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01P 3/00 - Fungicides

Abstract

The present invention discloses an oxime ether compound with a novel structure, wherein the structure is represented by general formula (I), and the definition of each substituent in the formula is described in the description. The compound of general formula (I) has excellent bactericidal activity, and exhibits a good prevention and control effect on plant bacterial diseases and fungal diseases, and included is a use of the compound of general formula (I) as a bactericide in agriculture and other fields.

IPC Classes  ?

• C07C 255/62 - Carboxylic acid nitriles containing cyano groups and oxygen atoms being part of oxyimino groups bound to the same carbon skeleton
• C07D 277/24 - Radicals substituted by oxygen atoms
• C07D 261/12 - Oxygen atoms
• A01N 43/76 - 1,3-OxazolesHydrogenated 1,3-oxazoles
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• A01P 3/00 - Fungicides

Abstract

Provided are a phenylisoxazoline compound and use thereof. The phenylisoxazoline compound is represented by general formula (I). The compound of general formula (I) has good herbicidal activity, and can effectively control barnyard grass, Setaria viridis, Cyperus difformis, Juncellus serotinus, Digitaria sanguinalis, Arthraxon hispidus, Abutilon theophrasti, Zinnia elegans, Amaranthus retroflexus, Portulaca oleracea, Xanthium strumarium, Solanum nigrum, Cassia tora, Hibiscus trionum, Glycine soja and other weeds; furthermore, the compound can obtain good weeding effect at low dosage, has certain safety to crops such as corn, wheat and rice, and can be used as a herbicide in agriculture.

IPC Classes  ?

• C07D 413/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 261/04 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
• C07D 471/04 - Ortho-condensed systems
• C07D 487/04 - Ortho-condensed systems
• C07D 513/04 - Ortho-condensed systems
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 43/50 - 1,3-DiazolesHydrogenated 1,3-diazoles
• A01N 43/653 - 1,2,4-TriazolesHydrogenated 1,2,4-triazoles
• A01N 43/836 - 1,2,4-Oxa(thia)diazolesHydrogenated 1,2,4-oxa(thia)diazoles
• A01N 47/12 - Carbamic acid derivatives, i.e. containing the group —O—CO—NThio-analogues thereof containing a —O—CO—N group, or a thio-analogue thereof, neither directly attached to a ring nor the nitrogen atom being a member of a heterocyclic ring
• A01N 55/10 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing silicon
• A01P 13/00 - HerbicidesAlgicides

Abstract

Disclosed is a piperidinamine compound containing fused ring pyrimidine, the structure of the compound being as shown in general formula L: the definition of each substituent in the formula is shown in the description. The compound of the present invention has broad-spectrum bactericidal activity, and has excellent pest control effects on cucumber downy mildew, wheat powdery mildew, corn rust, cucumber anthracnose, and so on. In addition, the compound of the present invention also exhibits good insecticidal and acaricidal activity, and has excellent pest control effects on Plutella xylostella, Leucania separata, Tetranychus cinnabarinus, and so on.

IPC Classes  ?

• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 239/46 - Two or more oxygen, sulfur or nitrogen atoms
• C07D 239/42 - One nitrogen atom
• C07D 239/52 - Two oxygen atoms
• C07D 495/04 - Ortho-condensed systems
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines

Abstract

An amide compound containing a substituted acetophenone structure fragment, having a structure shown as general formula I. Please see the description for the definitions of substituents in the formula. The compound has a broad-spectrum bactericidal activity, and has excellent prevention and treatment effects on cucumber downy mildew, wheat powdery mildew, corn rust, cucumber anthracnose, cucumber gray mold, tomato gray mold, etc.

IPC Classes  ?

• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01N 43/60 - 1,4-DiazinesHydrogenated 1,4-diazines
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 35/04 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having two bonds to hetero atoms with at the most one bond to halogen, e.g. aldehyde radical containing aldehyde or keto groups, or thio-analogues thereof, directly attached to an aromatic ring system, e.g. acetophenoneDerivatives thereof, e.g. acetals
• A01N 37/30 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N, e.g. carboxylic acid amides or imidesThio-analogues thereof containing the groups —CO—N and both being directly attached by their carbon atoms to the same carbon skeleton, e.g. H2N—NH—CO—C6H4—COOCH3Thio-analogues thereof
• C07D 231/10 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
• C07D 213/02 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
• C07D 239/24 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
• C07D 241/10 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
• C07D 275/02 - Heterocyclic compounds containing 1, 2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
• C07D 277/20 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members

Abstract

Provided is a pyrimidine-containing piperidinamine compound, the structure of which is shown in general formula I: the definition of each substituent in the formula is shown in the description. The provided compound shows good insecticidal and acaricidal activity, and has excellent pest control effects on Plutella xylostella, Tetranychus cinnabarinus, and so on. In addition, the described compound has broad-spectrum bactericidal activity, and has excellent pest control effects on cucumber downy mildew, wheat powdery mildew, cucumber anthracnose, and so on.

IPC Classes  ?

• C07D 239/46 - Two or more oxygen, sulfur or nitrogen atoms
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines

Abstract

The present invention relates to the field of insecticides and acaricides, and relates to a synergistic insecticidal and acaricidal composition. The composition contains active component A and active component B, and the ratio of the parts by weight of active component A to those of active component B is 1:99 to 99:1. Active component A is selected from compound I, and active component B is selected from fluazinam, bifenazate, chlorfenapyr, Pyflubumider, Acynonspy, a pyrethroid insecticide or a pyrethroid acaricide. The structure of active component A is as follows. The composition of the present invention has advantages such as obvious synergy and delayed resistance, and can be used for control a variety of pests.

IPC Classes  ?

• A01N 31/16 - Oxygen or sulfur directly attached to an aromatic ring system with two or more oxygen or sulfur atoms directly attached to the same aromatic ring system
• A01N 41/10 - SulfonesSulfoxides
• A01N 43/90 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
• A01N 43/22 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with one hetero atom rings with more than six members
• A01N 43/12 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with one hetero atom five-membered rings condensed with a carbocyclic ring
• A01N 47/38 - Ureas or thioureas containing the groups N—CO—N or N—CS—N containing the group N—CO—N where at least one nitrogen atom is part of a heterocyclic ringThio-analogues thereof
• A01N 47/34 - Ureas or thioureas containing the groups N—CO—N or N—CS—N containing the groups , e.g. biuretThio-analogues thereofUrea-aldehyde condensation products
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 47/24 - Carbamic acid derivatives, i.e. containing the group —O—CO—NThio-analogues thereof containing the groups , or Thio-analogues thereof
• A01N 37/42 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing within the same carbon skeleton a carboxylic group or a thio-analogue, or a derivative thereof, and a carbon atom having only two bonds to hetero atoms with at the most one bond to halogen, e.g. keto-carboxylic acids
• A01N 43/58 - 1,2-DiazinesHydrogenated 1,2-diazines
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides

Abstract

Provided are an isoxazoline compound of formula (I) having an optical activity and a use thereof, the compound of formula (I) has good herbicidal activity, can be used for pre-seedling and post-seedling weeding, and can also be used for soil treatment. Various broadleaf weeds and gramineous weeds as well as cyperaceae weeds can be effectively controlled, and various resistant weeds such as glyphosate resistant weeds can be prevented. The compound can obtain good weeding effects at low doses, and have good safety for crops such as corn, wheat, rice, soybean, beet and the like, can be used as a selective herbicide for crops in agriculture, and can also be used as a sterilant herbicide for non-cultivated/lobed land, forest land, orchard, ridge, etc.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention relates to the field of agricultural herbicides, and particularly relates to an isoxazoline compound with optical activity and the uses thereof. The isoxazoline compound with optical activity is shown in the formula (I). The compound of the formula (I) has excellent herbicidal activity, can be used for weeding pre- and post- emergence, and can also be used for soil treatment. The compound of the formula (I) can effectively control various broad-leaved weeds, grass weeds and Cyperaceae weeds, and can control various resistant weeds, such as glyphosate-resistant weeds. The excellent weeding effect can be obtained at a low dose. The compound has good safety to crops such as corn, wheat, rice, soybean and sugar beet. The compound can be used as a selective herbicide in crop fields in agriculture, and can also be used as a non-selective herbicide in non¬ cultivated land, fallow land, woodland, orchards and ridges.

IPC Classes  ?

• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

Disclosed herein is a herbicidal composition, comprising an active component A and an active component B, wherein the active component B is one selected from the group consisting of glufosinate-ammonium, glufosinate-P-ammonium, oxyfluorfen, acetoflufen, imazethapyr, dimethoxamide, dimethoxamid-P, metolachlor, S-metolachlor, butachlor, acetochlor, pyroxasulfone, glyphosate and derivatives thereof.

IPC Classes  ?

• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 25/04 - Dispersions or gels
• A01N 25/14 - Powders or granules wettable
• A01N 33/22 - Nitro compounds containing oxygen or sulfur attached to the carbon skeleton containing the nitro group having at least one oxygen or sulfur atom and at least one nitro group directly attached to the same aromatic ring system
• A01N 37/22 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N, e.g. carboxylic acid amides or imidesThio-analogues thereof the nitrogen atom being directly attached to an aromatic ring system, e.g. anilides
• A01N 43/10 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with one hetero atom five-membered rings with sulfur as the ring hetero atom
• A01N 43/50 - 1,3-DiazolesHydrogenated 1,3-diazoles
• A01N 57/20 - Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-carbon bonds containing acyclic or cycloaliphatic radicals

Abstract

The present invention discloses an alkene-containing carboxylic ester compound and an application of agriculturally acceptable salt as a herbicide. The compound is shown in formula (I). The definition of each substituent in the formula I is described in the description. The compound of the formula I of the present invention has excellent herbicidal activity and can be used for controlling agricultural weeds.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01N 43/653 - 1,2,4-TriazolesHydrogenated 1,2,4-triazoles
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• C07D 231/20 - One oxygen atom attached in position 3 or 5
• C07D 401/06 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• C07D 403/10 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

Disclosed are an alkene-containing amide compound and the use of an agriculturally acceptable salt thereof as a herbicide. The compound is as represented by general formula (I): the substituents in general formula I are defined in the description. The compound of general formula I of the present invention has an excellent herbicidal activity and can be used to control agricultural weeds.

IPC Classes  ?

• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 43/836 - 1,2,4-Oxa(thia)diazolesHydrogenated 1,2,4-oxa(thia)diazoles
• C07D 257/06 - Five-membered rings with nitrogen atoms directly attached to the ring carbon atom
• C07D 285/08 - 1,2,4-ThiadiazolesHydrogenated 1,2,4-thiadiazoles
• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 405/12 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 413/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Disclosed in the present invention are a carboxylic acid ester compound and an application thereof, the structure of the compound being shown in general formula I, and the definition of each substituent in general formula I being provided in the specification. The compound of general formula I has excellent herbicidal activity and can be used for the prevention and control of agricultural weeds.

IPC Classes  ?

• C07D 231/20 - One oxygen atom attached in position 3 or 5
• C07D 407/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• A01N 43/48 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

Disclosed are an alkene-containing amide compound and the use of an agriculturally acceptable salt thereof as a herbicide. The compound is as represented by general formula (I): the substituents in general formula I are defined in the description. The compound of general formula I of the present invention has an excellent herbicidal activity and can be used to control agricultural weeds.

IPC Classes  ?

• C07D 257/06 - Five-membered rings with nitrogen atoms directly attached to the ring carbon atom
• C07D 405/12 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 285/08 - 1,2,4-ThiadiazolesHydrogenated 1,2,4-thiadiazoles
• C07D 413/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/713 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
• A01N 43/836 - 1,2,4-Oxa(thia)diazolesHydrogenated 1,2,4-oxa(thia)diazoles
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

Disclosed in the present invention are an alkene-containing carboxylate compound and use of an agriculturally acceptable salt thereof as a herbicide. Said compound is as represented by general formula (I). The definition of the substituents in general formula I is shown in the description. The compound of general formula I of the present invention has an excellent herbicidal activity, and can be used for preventing and treating agricultural weeds.

IPC Classes  ?

• C07D 231/20 - One oxygen atom attached in position 3 or 5
• C07D 401/06 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
• C07D 403/10 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 43/653 - 1,2,4-TriazolesHydrogenated 1,2,4-triazoles

Abstract

The present invention relates to the field of insecticides and acaricides, and in particular, to a piperic acid derivative and an application thereof. The structure is as shown in general forrnula l , and the definition of each substituent in the formula is as described in the specification. A compound of formula l has excellent insecticidal and acaricidal activities and can be used for preventing various pests and mites. (l)

IPC Classes  ?

• A01N 43/30 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with two or more hetero atoms five-membered rings with two hetero atoms in positions 1,3 with two oxygen atoms in positions 1,3, condensed with a carbocyclic ring
• C07D 317/46 - Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Abstract

The present invention relates to the field of insecticides and acaricides, and in particular, to a piperic acid derivative and an application thereof. The structure is as shown in general formula I, and the definition of each substituent in the formula is as described in the specification. A compound of formula I has excellent insecticidal and acaricidal activities and can be used for preventing various pests and mites.

IPC Classes  ?

• C07D 317/46 - Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
• A01N 43/30 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with two or more hetero atoms five-membered rings with two hetero atoms in positions 1,3 with two oxygen atoms in positions 1,3, condensed with a carbocyclic ring

Abstract

Disclosed are a carboxylic acid oxime ester compound and the use thereof as a herbicide and for preparing a microbicide. The carboxylic acid oxime ester compound is as represented by general formula I:

IPC Classes  ?

• C07C 233/75 - Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
• C07C 251/68 - Oximes having oxygen atoms of oxyimino groups esterified by carboxylic acids with at least one of the esterifying carboxyl groups bound to a carbon atom of a six-membered aromatic ring
• C07C 251/44 - Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups being part of a ring other than a six-membered aromatic ring
• C07D 231/14 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention relates to a fungicidal and bactericidal composition and an application method therefor. The composition comprises two active components A and B, wherein component A is selected from compounds represented by general formula I, and component B is selected from a succinate dehydrogenase inhibitor microbicide, a copper-containing microbicide, an antibiotic compound, an antibiotic compound salt or zinc thiazole. The weight ratio of the two active components of the composition is from 1:100 to 100:1. The composition of the present invention is used to prevent various plant diseases caused by pathogenic fungi and bacteria.

IPC Classes  ?

• A01N 37/50 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio-analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio-analogue of a carboxylic group, e.g. amino-carboxylic acids the nitrogen atom being doubly bound to the carbon skeleton
• A01N 47/40 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
• A01N 37/34 - Nitriles
• A01N 37/48 - Nitro-carboxylic acidsDerivatives thereof
• A01P 3/00 - Fungicides

Abstract

The present invention relates to a stable herbicide composition, the composition comprising active ingredients A and B. The component A is selected from a compound represented by the following general formula (I). The component B is selected from glyphosate and suitable salts or esters thereof. When a solid preparation is prepared, the active component A is first adsorbed using an adsorption carrier, and an adsorption product is then mixed with the component B, promoter, and filler to obtain a stable solid preparation.

IPC Classes  ?

• A01N 57/20 - Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-carbon bonds containing acyclic or cycloaliphatic radicals
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 25/22 - Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of applicationSubstances for reducing the noxious effect of the active ingredients to organisms other than pests containing ingredients stabilising the active ingredients
• A01P 13/00 - HerbicidesAlgicides

Abstract

A pyrazole amide compound and an application thereof as a herbicide. The compound is as represented by formula (I). The compound as represented by formula (I) has herbicidal activity and can be used for controlling agricultural weeds.

IPC Classes  ?

• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 405/14 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
• C07D 413/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
• C07D 403/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• A01N 43/713 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention relates to a stable herbicide composition, the composition comprising active ingredients A and B. The component A is selected from a compound represented by the following general formula (I). The component B is selected from glyphosate and suitable salts or esters thereof. When a solid preparation is prepared, the active component A is first adsorbed using an adsorption carrier, and an adsorption product is then mixed with the component B, promoter, and filler to obtain a stable solid preparation.

IPC Classes  ?

• A01N 25/22 - Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of applicationSubstances for reducing the noxious effect of the active ingredients to organisms other than pests containing ingredients stabilising the active ingredients
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01N 57/20 - Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-carbon bonds containing acyclic or cycloaliphatic radicals
• A01P 13/00 - HerbicidesAlgicides

Abstract

Disclosed are a herbicide composition and an application method thereof. The composition comprises active component A and active component B, wherein component A is selected from compounds of Formula (I), and component B is selected from diquat. The herbicide composition is particularly suitable for preventing and weeding weeds that are resistant to organophosphorus herbicides, particularly glyphosate.

IPC Classes  ?

• A01N 43/90 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

A method for preparing a sulfur-containing biphenyl compound as shown in the general formula (I), the reaction formula aa being as shown in the specification. The method for coupling reaction under the combined action of metal and zinc uses halogenated benzene as shown in the general formula (II), and a catalyst system composed of a nickel compound and at least one ligand so as to obtain the sulfur-containing biphenyl compound shown in the general formula (I).

IPC Classes  ?

• C07C 319/20 - Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by reactions not involving the formation of sulfide groups
• C07C 323/09 - Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton

Abstract

The present invention belongs to the field of organic synthesis, in particular relates to a method for preparing an isoxazoline-containing uracil compound by methylation. The isoxazoline-containing uracil compound shown by formula (I) is prepared by a methylation reaction of a compound shown by formula (II) and monochloromethane in a closed container in the presence of an alkali, a catalyst and an organic solvent, the reaction equation therefor is as follows and the definition of each group in the formula is as in the description. The preparation method provided by the present invention can avoid harm possibly brought by the use of methyl iodide, is safe and environmentally friendly, has a low cost and a high product content, and is suitable for industrialization.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

The present invention belongs to the field of organic synthesis, in particular relates to a method for preparing an isoxazoline-containing uracil compound by methylation. The isoxazoline-containing uracil compound shown by formula (I) is prepared by a methylation reaction of a compound shown by formula (II) and monochloromethane in a closed container in the presence of an alkali, a catalyst and an organic solvent, the reaction equation therefor is as follows and the definition of each group in the formula is as in the description. The preparation method provided by the present invention can avoid harm possibly brought by the use of methyl iodide, is safe and environmentally friendly, has a low cost and a high product content, and is suitable for industrialization.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

The present invention belongs to the field of acaricides, and relates to a biphenyl compound-containing liquid preparation and an application thereof. The biphenyl compound-containing liquid preparation uses compound A as an active component, mixed with at least one carrier and at least one auxiliary agent, the weight percentage of the active component of the liquid preparation being 0.1-99%. The liquid preparation of the present invention allows the particle size of the liquid preparation to be controlled by a good auxiliary agent system, and the liquid preparation has features such as good dispersibility, high suspension rate, high biological activity, small dosage, low cost, resistance to rain erosion, low residue, and low toxicity to humans and animals.

IPC Classes  ?

• A01N 31/16 - Oxygen or sulfur directly attached to an aromatic ring system with two or more oxygen or sulfur atoms directly attached to the same aromatic ring system
• A01N 41/10 - SulfonesSulfoxides
• A01N 25/02 - Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of applicationSubstances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
• A01P 7/02 - Acaricides

Abstract

Provided are a method for preparing a propanedinitrile oxime ether compound and an intermediate compound. The propanedinitrile oxime ether compound has a structure as shown in formula (VII), wherein W is selected from aryl or heteroaryl. The preparation method comprises: reacting a first raw material with a second raw material under the action of a first solvent and a catalyst to obtain an intermediate compound, wherein the first raw material has a structure as shown in formula (IV), and the second raw material has a structure as shown in formula (V); and subjecting the intermediate compound as shown in formula (VI) and a dehydrant to a dehydration reaction under the action of a second solvent to obtain the propanedinitrile oxime ether compound. In the preparation process for the intermediate, a cheaper cyanoacetamide is used as a raw material, and the reaction conditions are mild. Moreover, the yield of the intermediate compound is high and the cost of the process is low. Furthermore, the desired propanedinitrile oxime ether compound is obtained only through a one-step dehydration reaction. Using the preparation method is advantageous for improving the yield of the propanedinitrile oxime ether and reducing the cost of the process.

IPC Classes  ?

• C07C 253/20 - Preparation of carboxylic acid nitriles by dehydratation of carboxylic acid amides
• C07C 255/64 - Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton with the nitrogen atoms further bound to oxygen atoms
• C07C 253/30 - Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
• C07D 277/24 - Radicals substituted by oxygen atoms
• C07D 213/61 - Halogen atoms or nitro radicals
• C07D 277/32 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 215/14 - Radicals substituted by oxygen atoms

Abstract

Disclosed is a substituted pyrimidine compound. The structure of same is as shown in formula I; and for the definitions of each substituent see the description. The compound of the present invention has broad-spectrum fungicidal, insecticidal and acaricidal activities, and has excellent prevention and control effects on cucumber downy mildew, powdery mildew, corn rust, anthracnose, rice blast, aphids and Tetranychus cinnabarinus, etc. (I)

IPC Classes  ?

• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• C07D 417/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• A01P 3/00 - Fungicides
• A01P 7/04 - Insecticides
• A01P 7/02 - Acaricides
• A01P 5/00 - Nematocides

Abstract

The present invention provides a polymorph of a benzamide compound and a preparation method and applications thereof. The shown benzamide compound is 3-Bromo-N-[2,4-dichloro-6-[(methylamino)carbonyl]phenyl]-1-(3,5-dichloro-2-pyridinyl)-1H-pyrazole-5-carboxamide. The application of the polymorph of the compound in the preparation of the formulation exhibits excellent effect. The advantages of the polymorph A in aspects such as chemical stability, filterability, solubility, hygroscopicity, melting point, solid density and flowability can have a significant impact on the developments of the production method and a formulation and on the quality and efficacy of a plant treating agent.

IPC Classes  ?

• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond

Abstract

A piperic acid derivative and preparation and an application thereof. The structure of the derivative is as shown in general formula I. The compound of general formula I has excellent pesticidal, miticidal, and bactericidal activities and can be used in preventing various pests, pest mites, or harmful bacteria.

IPC Classes  ?

• C07C 237/42 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
• C07C 323/42 - Y being a carbon atom of a six-membered aromatic ring
• C07D 231/12 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
• C07D 261/18 - Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
• A01N 37/22 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N, e.g. carboxylic acid amides or imidesThio-analogues thereof the nitrogen atom being directly attached to an aromatic ring system, e.g. anilides
• A01N 43/36 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings

Abstract

Disclosed is a malononitrile oxime ether compound having a novel structure as shown in the general formula I. Respective substituents in the general formula I as defined in the specification. The compound of the general formula I exhibits an excellent microbicidal activity, and can effectively prevent and treat plant diseases caused by bacteria and fungi. Also provided is a use of the compound of the general formula I as a microbicide in the agricultural and other fields.

IPC Classes  ?

• A01N 33/24 - Biocides, pest repellants or attractants, or plant growth regulators containing organic nitrogen compounds containing nitrogen-to-oxygen bonds only one oxygen atom attached to the nitrogen atom
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• C07C 255/64 - Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton with the nitrogen atoms further bound to oxygen atoms
• C07C 251/58 - Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals of hydrocarbon radicals substituted by nitrogen atoms not being part of nitro or nitroso groups
• C07C 251/56 - Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals of hydrocarbon radicals substituted by doubly-bound oxygen atoms
• C07C 251/54 - Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals of hydrocarbon radicals substituted by singly-bound oxygen atoms
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 43/42 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 213/61 - Halogen atoms or nitro radicals
• C07D 215/14 - Radicals substituted by oxygen atoms
• C07D 231/12 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
• C07D 231/14 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 277/28 - Radicals substituted by nitrogen atoms
• C07D 277/64 - Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2

Abstract

Echinochloa crusgalli, Setaria viridis, Cyperus difformis, Juncellus serotinus, Digitaria sangunalis, Arthraxon hispidus, Abutilon theophrasti, Zinnia elegans, Amaranthus retrofluxes, Portulaca oleracea, Xanthium sibiricum, Solanum nigrum, Cassia tora, Hibiscus trionum, Glycine soja, an so on. They can effectively control weeds even at lower doses. The present invention compounds also safe to wheats, corns and rices, and can used as herbicides in agriculture fields.

IPC Classes  ?

• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• C07D 413/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Abstract

Disclosed are substituted pyrazole compounds containing pyrimidinyl as shown in Formula I: The definitions of each of the substituents can be seen in the description. The compounds of present invention have a good spectrum of bactericidal, insecticidal and acaricidal activity, and have good control effect on downy mildew of cucumber, powdery mildew of wheat, corn rust, rice blast, cucumber anthracnosis and the like. The compounds of present invention also show good insecticidal activity.

IPC Classes  ?

• C07D 513/04 - Ortho-condensed systems
• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• C07D 495/04 - Ortho-condensed systems
• C07D 417/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 239/72 - QuinazolinesHydrogenated quinazolines
• C07D 403/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• C07D 409/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
• C07D 487/04 - Ortho-condensed systems
• C07D 498/04 - Ortho-condensed systems

Abstract

Disclosed in the present invention is a pyridazinone compound having the structure as shown in general formula I, the definition of each substituent in the formula is described in the description. The compound of the present invention has broad-spectrum bactericidal, insecticidal and acaricidal activities, and has excellent prevention and control effects on cucumber downy mildew, wheat powdery mildew, corn rust, rice blast and cucumber anthracnose and the like.

IPC Classes  ?

• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/58 - 1,2-DiazinesHydrogenated 1,2-diazines
• A01P 3/00 - Fungicides
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides

Abstract

The present invention belongs to the field of fungicides, and relates to an amide compound and the preparation method and use thereof. The amide compound is as shown in general formula I: Each substituent in Formula I is defined in the description. The compound of general formula I of the present invention has an outstanding fungicidal activity, and can be used for controlling fungal diseases.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 231/16 - Halogen atoms or nitro radicals
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• C07D 231/14 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 277/56 - Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Abstract

Provided are a polymorph of a benzamide compound and a preparation method and a use thereof. The shown benzamide compound is 3-bromo-1-(3,5-dichloro-2-pyridyl)-N-[2,4-dichloro-6-[(methylamino)carbonyl]phenyl]-1H-pyrazole-5-methanamide. A polymorph of the compound exhibits an excellent effect in aspects such as the use in preparing a preparation. The advantages of the polymorph A in aspects such as chemical stability, filterability, solubility, hygroscopicity, melting point, solid density and flowability can have a significant impact on the developments of the production method and a preparation and on the quality and efficacy of a plant treating agent.

IPC Classes  ?

• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01P 7/04 - Insecticides
• A01P 3/00 - Fungicides

Abstract

The present disclosure relates to acaricide, specifically to a kind of biphenyl compounds and uses thereof. The general formula I is as follows: wherein: each substituent is defined as that in the description. The compounds of the general formula I show high acaricidal activities and can be used for controlling various harmful mites.

IPC Classes  ?

• C07C 323/09 - Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
• A01N 31/08 - Oxygen or sulfur directly attached to an aromatic ring system
• C07C 317/12 - SulfonesSulfoxides having sulfone or sulfoxide groups bound to carbon atoms of rings other than six-membered aromatic rings

Abstract

The present invention belongs to the field of organic synthesis, and in particular relates to a method for preparing a pyridylpyrazolidone carboxylate compound. The reaction formula is as follows and the definition for each group in the formula can be found in the description. The present invention provides a method for preparing a pyridylpyrazolidone carboxylate compound that is a key intermediate of benzamide insecticides. By employing the method of the present invention, the yield of products is increased, and the energy consumption is reduced. The method of the present invention is more easily to be used in the industrial production.

IPC Classes  ?

• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond

Abstract

Disclosed is a malononitrile oxime ether compound having a novel structure as shown in the general formula I. Respective substituents in the general formula I are as defined in the specification. The compound of the general formula I exhibits an excellent microbicidal activity, and can effectively prevent and treat plant diseases caused by bacteria and fungi. Also provided is a use of the compound of the general formula I as a microbicide in the agricultural and other fields.

IPC Classes  ?

• C07C 255/64 - Carboxylic acid nitriles containing cyano groups and nitrogen atoms further bound to other hetero atoms, other than oxygen atoms of nitro or nitroso groups, bound to the same carbon skeleton with the nitrogen atoms further bound to oxygen atoms

Abstract

The invention relates to the field of mite killers, and specifically, to a biphenyl compound and application thereof. The structure is expressed by formula I, and each substituent in the formula is defined in the specification. The formula I compound has favorable acaricidal activity, and can be used in preventing and treating all kinds of mite problems.

IPC Classes  ?

• C07C 323/09 - Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
• C07C 317/14 - SulfonesSulfoxides having sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings
• A01N 31/16 - Oxygen or sulfur directly attached to an aromatic ring system with two or more oxygen or sulfur atoms directly attached to the same aromatic ring system
• A01N 41/10 - SulfonesSulfoxides

Abstract

Provided are an unsaturated oximino ether compound and a use thereof. The compound is as shown by general formula I, wherein the compound of formula I has an excellent bactericidal activity, and especially still has good control effect on cucumber downy mildew and wheat powdery mildew at a relatively low dose, while also having an excellent systemic action. Therefore, the compound as shown by general formula I is used as a bactericide in the agricultural and other fields.

IPC Classes  ?

• C07C 251/60 - Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals of hydrocarbon radicals substituted by carboxyl groups
• A01N 37/36 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio-analogue, or a derivative thereof, and a singly bound oxygen or sulfur atom attached to the same carbon skeleton, this oxygen or sulfur atom not being a member of a carboxylic group or of a thio-analogue, or of a derivative thereof, e.g. hydroxy-carboxylic acids
• A01N 37/50 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio-analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio-analogue of a carboxylic group, e.g. amino-carboxylic acids the nitrogen atom being doubly bound to the carbon skeleton

Abstract

Disclosed is a substituted pyrazole compound containing pyrimidine, wherein the structure is as shown in formula (I). See the description for the definition of each substituent. The compound of the present invention has a broad-spectrum fungicidal, insecticidal and acaricidal activity, and has a good controlling effect on cucumber downy mildew, wheat powdery mildew, corn rust, rice blast, cucumber anthracnose, etc. The compound of the present invention also exhibits a good insecticidal activity.

IPC Classes  ?

• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 495/04 - Ortho-condensed systems
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• A01P 3/00 - Fungicides
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides
• A01P 1/00 - DisinfectantsAntimicrobial compounds or mixtures thereof
• A01P 5/00 - Nematocides

Abstract

Disclosed is a substituted pyrazole compound containing pyrimidine, wherein the structure is as shown in formula (I). See the description for the definition of each substituent. The compound of the present invention has a broad-spectrum fungicidal, insecticidal and acaricidal activity, and has a good controlling effect on cucumber downy mildew, wheat powdery mildew, corn rust, rice blast, cucumber anthracnose, etc. The compound of the present invention also exhibits a good insecticidal activity.

IPC Classes  ?

• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• A01P 1/00 - DisinfectantsAntimicrobial compounds or mixtures thereof
• A01P 3/00 - Fungicides
• A01P 5/00 - Nematocides
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides
• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 495/04 - Ortho-condensed systems

Abstract

Disclosed are pyrazolyl pyrimidinamine compounds with structures as shown in Formula I: The definitions of each of the substituents can be seen in the description. Myzus persicae, Tetranychus cinnabarinus etc.

IPC Classes  ?

• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 403/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• C07D 417/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings

Abstract

The present invention belongs to the field of fungicides, and relates to an amide compound and the preparation method and use thereof. The amide compound is as shown in general formula I: each substituent in general formula I is defined in the description. The compound of general formula I of the present invention has an outstanding fungicidal activity, and can be used for controlling fungal diseases.

IPC Classes  ?

• C07D 231/14 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 277/56 - Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01P 3/00 - Fungicides

Abstract

Disclosed is a pyrazole amide compound of a novel structure as represented by general formula I, wherein, each substituent group is as defined in the specification. The compound of general formula I has good insecticidal activity, and can be used for pest control.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Abstract

The present invention belongs to the field of agricultural herbicides, and in particular relates to a pyrimidine urea compound containing isoxazolines and a use thereof. The pyrimidine urea compound containing isoxazolines is as shown in general formula (I). The compounds of general formula (I) have a very good herbicidal activity, and can effectively control barnyard grass, green bristlegrass, Cyperus difformis, Juncellus serotinus, Digitaria sanguinalis, Arthraxon hispidus, Abutilon theophrasti, Zinnia elegans, Amaranthus retroflexus, purslane, Xanthium sibiricum, Solanum nigrum,Senna obtusifolia, Hibiscus trionum, Glycine ussuriensis, and the like, and can obtain a very good herbicidal effect at low doses, is relatively safe for crops such as corn, wheat and rice, and can be used as a herbicide in agriculture.

IPC Classes  ?

• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides

Abstract

The present invention belongs to the field of agricultural herbicides, and in particular relates to a pyrimidine urea compound containing isoxazolines and a use thereof. The pyrimidine urea compound containing isoxazolines is as shown in general formula (I). The compounds of general formula (I) have a very good herbicidal activity, and can effectively control barnyard grass, green bristlegrass, Cyperus difformis, Juncellus serotinus, Digitaria sanguinalis, Arthraxon hispidus, Abutilon theophrasti, Zinnia elegans,Amaranthus retroflexus, purslane, Xanthium sibiricum, Solanum nigrum,Senna obtusifolia, Hibiscus trionum, Glycine ussuriensis,and the like, and can obtain a very good herbicidal effect at low doses, is relatively safe for crops such as corn, wheat and rice, and can be used as a herbicide in agriculture.

IPC Classes  ?

• A01N 43/80 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
• A01P 13/00 - HerbicidesAlgicides
• C07D 413/10 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

Disclosed is a substituted pyrimidine compound having a structure as represented by formula PY. See the description for the definition of each substituent in the formula. The compound of the present invention provides broad-spectrum bactericidal, pesticidal, and acaricidal activities, provides great control effects against plant diseases such as cucumber downy mildew, corn rust, wheat powdery mildew, rice blast, and cucumber gray mold, specifically provides improved control effects against cucumber downy mildew, corn rust, wheat powdery mildew, and rice blast, provides great control effects against aphid, carmine spider mite, diamondback moth, and armyworm, and acquires great effects at a minimal dosage. The compound of the present invention also provides characteristics such as a simplified preparation method.

IPC Classes  ?

• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• A01N 43/58 - 1,2-DiazinesHydrogenated 1,2-diazines
• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 403/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• C07D 239/28 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
• C07D 253/07 - 1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 239/42 - One nitrogen atom

Abstract

The invention discloses a homopiperony lamine compound which has a structural general formula I as follows as shown in the specification: wherein definitions of substituents in the formula are as shown in the specification. tetranychus cinabarinus boisdu.

IPC Classes  ?

• A61K 31/506 - PyrimidinesHydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
• C07D 239/42 - One nitrogen atom
• C07D 317/50 - Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
• C07D 405/12 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 405/14 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• C07D 409/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
• C07D 417/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings

Abstract

Disclosed are pyrazolyl pyrimidinamine compounds with structures as shown in Formula I. The definitions of each of the substituents can be seen in the description. The compounds of present invention have a broad spectrum of bactericidal, insecticidal and acaricidal activity, and have good control effect on downy mildew of cucumber, powdery mildew of wheat, corn rust, anthracnosis of cucumber and the like, and especially have better control effect on downy mildew of cucumber, powdery mildew of wheat and anthracnosis of cucumber. The compounds of present invention also show good insecticidal activity, part of the compounds, at very low doses, have excellent control effect on diseases caused by Plutella xylostella, armyworm, Myzus persicae, Tetranychus cinnabarinus etc.

IPC Classes  ?

• C07D 403/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• C07D 417/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• A01P 3/00 - Fungicides
• A01P 7/04 - Insecticides
• A01P 7/02 - Acaricides
• A01P 5/00 - Nematocides

Abstract

Disclosed is a pyrazole amide compound of a novel structure as represented by general formula I, wherein, each substituent group is as defined in the specification. The compound of general formula I has good insecticidal activity, and can be used for pest control.

IPC Classes  ?

• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01P 7/04 - Insecticides

Abstract

Disclosed is a pyrazole amide compound as represented by general formula I, wherein, R1 is selected from hydrogen, C1-C4 alkyl, C2-C6 alkenyl, and C1-C6 alkyl; and R2 and R3 can be the same or different, and are respectively and independently selected from the C1-C6 alkyl. The general formula I compound has an excellent bactericidal activity, and can be used to prevent and control fungal diseases.

IPC Classes  ?

• C07D 231/14 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01P 3/00 - Fungicides

Abstract

Disclosed in the present invention is aryl pyridine (pyrimidine) compound having a structure as shown by the general formula (I) below, wherein the substituents in the formula are as defined in the description. The compound of formula I displays relatively high activities on harmful insects, mites and eggs in the fields of agriculture, and civil and animal technology, especially having better activities on harmful mites such as Tetranychus cinnabarinus etc., and can obtain very good effects at a very low dose.

IPC Classes  ?

• C07D 213/85 - Nitriles in position 3
• A01N 43/60 - 1,4-DiazinesHydrogenated 1,4-diazines
• A01P 7/02 - Acaricides

Abstract

Disclosed is a substituted cyanoaniline compound or a salt thereof, wherein the compound has a structure represented by General Formula I. The compound of General Formula I has broad-spectrum fungicidal activity in the field of agriculture and effectively prevents against a variety of pathogens such as cucumber downy mildew, wheat powdery mildew, maize rust disease, rice blast and cucumber gray mold. In particular, even at a low dose, the compound effectively prevents and treats rice blast, cucumber gray mold, maize rust disease and cucumber downy mildew. Moreover, the raw materials for preparing the compounds are widely available and the synthesis method therefor is simple and convenient.

IPC Classes  ?

• A61K 31/495 - Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
• C07D 237/12 - Halogen atoms or nitro radicals
• A01N 37/34 - Nitriles
• A01N 59/04 - Carbon disulfideCarbon monoxideCarbon dioxide
• C07D 213/74 - Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
• C07C 255/58 - Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
• C07D 237/24 - Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
• C07D 239/52 - Two oxygen atoms
• C07D 241/26 - Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms
• C07C 255/59 - Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton the carbon skeleton being further substituted by singly-bound oxygen atoms
• C07C 255/60 - Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
• A01N 37/44 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio-analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio-analogue of a carboxylic group, e.g. amino-carboxylic acids
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• A01N 43/58 - 1,2-DiazinesHydrogenated 1,2-diazines
• A01N 43/60 - 1,4-DiazinesHydrogenated 1,4-diazines

Abstract

The present invention discloses an aryloxy dihalopropenyl ether compound with the structure shown as general formula (I), of which the group definitions can be seen in the specification. The present invention also discloses the use of the compound with general formula (I) as an insecticide in the agricultural field and an insecticidal composition using the compound with general formula (I) as an active component.

IPC Classes  ?

• A61K 31/395 - Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
• C07D 213/60 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• C07C 43/225 - Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring containing halogen
• C07C 43/29 - Ethers having an ether-oxygen atom bound to carbon atoms both belonging to six-membered aromatic rings containing halogen
• A01N 31/16 - Oxygen or sulfur directly attached to an aromatic ring system with two or more oxygen or sulfur atoms directly attached to the same aromatic ring system
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 43/58 - 1,2-DiazinesHydrogenated 1,2-diazines
• A01N 43/76 - 1,3-OxazolesHydrogenated 1,3-oxazoles
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 237/16 - Two oxygen atoms
• C07D 263/58 - BenzoxazolesHydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
• C07D 277/32 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 213/643 - 2-PhenoxypyridinesDerivatives thereof
• A01N 43/08 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with one hetero atom five-membered rings with oxygen as the ring hetero atom
• A01N 43/10 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atom with one hetero atom five-membered rings with sulfur as the ring hetero atom
• A01N 43/36 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
• A01N 43/50 - 1,3-DiazolesHydrogenated 1,3-diazoles
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• A01N 43/60 - 1,4-DiazinesHydrogenated 1,4-diazines

Abstract

The invention relates to substituted pyrimidine ammonia compounds. The structure of the compounds is represented as the general formula (I): The groups are as defined as specification. The compound represented by formula (I) can be used in the prevention of plants diseases caused by a plurality of pathogenic bacteria such as oomycota, basidiomycota, ascomycota, and fungi imperfecti, and due to these compounds have good bioactivity, which make them have very good effects at very low doses, especially more effective to powdery mildew of wheat. Therefore, the present invention relates to the use of the compounds having general formula I as fungicides, both in agriculture and other fields.

IPC Classes  ?

• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines
• A01N 47/06 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom containing —O—CO—O— groupsThio-analogues thereof
• C07D 239/47 - One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
• C07D 239/70 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
• C07D 405/12 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Substituted diphenylamine compounds of general formula I are provided, in which each substituted group is defined as in the description. The compounds of general formula I have broad-spectrum fungicidal activity in the field of agriculture. Furthermore, the preparation methods of the above compounds are simple.

IPC Classes  ?

• C07D 213/643 - 2-PhenoxypyridinesDerivatives thereof
• C07D 213/70 - Sulfur atoms
• C07C 211/56 - Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to two or three six-membered aromatic rings the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
• A01N 33/18 - Nitro compounds
• A01N 37/34 - Nitriles
• A01N 37/44 - Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio-analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio-analogue of a carboxylic group, e.g. amino-carboxylic acids
• A01N 41/10 - SulfonesSulfoxides
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• C07C 237/30 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having the nitrogen atom of the carboxamide group bound to hydrogen atoms or to acyclic carbon atoms
• C07C 237/40 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having the nitrogen atom of the carboxamide group bound to a carbon atom of a six-membered aromatic ring
• C07C 255/58 - Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
• C07C 317/36 - SulfonesSulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring with the nitrogen atoms of the amino groups bound to hydrogen atoms or to carbon atoms
• C07C 323/36 - Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton having at least one of the nitrogen atoms bound to a carbon atom of the same non-condensed six-membered aromatic ring the thio group being a sulfide group the sulfur atom of the sulfide group being further bound to an acyclic carbon atom
• C07C 327/48 - Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to carbon atoms of six-membered aromatic rings
• A01N 33/22 - Nitro compounds containing oxygen or sulfur attached to the carbon skeleton containing the nitro group having at least one oxygen or sulfur atom and at least one nitro group directly attached to the same aromatic ring system

Abstract

A kind of pyrazolyl acrylniitrile compounds represented by the structures of formula I or stereoisomers thereof are disclosed in the present invention. 2 or halogen. Or its stereoisomers. The Formula I compounds have high insecticidal activities or acaricidal activities, so they can be used as insecticide or acaricide.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 231/12 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Abstract

Tetranychus cinnabarinus, Tetranychidae, and the like. The said compounds show more excellent performance on inhibiting the incubation of eggs of harmful mites. The uses of the said compounds as insecticides and/or acaricides in agricultural and other fields also are disclosed.

IPC Classes  ?

• C07D 239/47 - One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
• A01N 43/54 - 1,3-DiazinesHydrogenated 1,3-diazines