Abstract

Disclosed in the present invention are an m-amidobenzoic acid bisamide compound as shown in formula (I) and intermediates thereof as shown in formulas (II) and (III), and a preparation method therefor and the use thereof, wherein substituents in the formulas are as defined in the description. The compound of the present invention has good insecticidal/acaricidal bioactivity and can be used for preventing and treating various pests and mites.

IPC Classes  ?

• C07D 213/82 - AmidesImides in position 3
• C07C 239/18 - Hydroxylamino compounds or their ethers or esters having nitrogen atoms of hydroxylamino groups further bound to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 53/00 - Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
• A01N 47/24 - Carbamic acid derivatives, i.e. containing the group —O—CO—NThio-analogues thereof containing the groups , or Thio-analogues thereof
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides
• A01G 13/00 - Protection of plants

Abstract

This invention provides 1-pyridyl pyrazole amide compounds represented by Formula (I) and preparation and uses thereof, wherein each substituent is defined in the disclosure. The compounds of Formula (I) of this invention possess excellent insecticidal activities, especially very strong activities against pests such as aphids, armyworms and diamondback moths, etc., and can be used to control various pests. This invention also provides synthetic intermediates represented by Formula (II) for preparing compounds of Formula (I) wherein each substituent is defined in the specification. This invention provides 1-pyridyl pyrazole amide compounds represented by Formula (I) and preparation and uses thereof, wherein each substituent is defined in the disclosure. The compounds of Formula (I) of this invention possess excellent insecticidal activities, especially very strong activities against pests such as aphids, armyworms and diamondback moths, etc., and can be used to control various pests. This invention also provides synthetic intermediates represented by Formula (II) for preparing compounds of Formula (I) wherein each substituent is defined in the specification.

IPC Classes  ?

• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond
• A01P 7/04 - Insecticides

Abstract

The present invention discloses a 1-pyridylpyrazole amide compound represented by formula (I), the preparation method and application thereof, and each substituent in the formula has the definition given by the description. The compound of formula (I) of the present invention has excellent insecticidal biological activity, especially high activity against pests such as aphids, armyworm and diamondback moth, and can be used to prevent and control various types of insect pests. The technical solution of the present invention also includes an intermediate for preparing the compound of formula (I), the structure of the intermediate is shown by the general formula (II), the definition of each substituent in the formula is shown in the description.

IPC Classes  ?

• C07D 401/04 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring- member bond
• C07C 211/46 - Aniline
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01P 7/00 - Arthropodicides

Abstract

Disclosed are pyridine sulfone as represented in formula (I) and derivatives of pyridine sulfone, and preparation method and application of pyridine sulfone. In formula (I), n, m, R, R1, R2, R3, R4, and R5 have the definitions given in the description. Formula (I) compound in the present invention has broad spectrum biological activities such as bactericidal and/or insecticidal/mite activities, especially has activities for diseases such as rice sheath blight and corn rust.

IPC Classes  ?

• C07D 213/61 - Halogen atoms or nitro radicals
• C07D 213/70 - Sulfur atoms
• C07D 213/74 - Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings

Abstract

Disclosed are thiazole methylamino pyridine compounds represented by the general formula (I) having fungicidal, insecticidal/acaricidal, and herbicidal activity, the preparation method thereof, the fungicidal, insecticidal/acaricidal, and herbicidal compositions containing the compounds of the present invention, and the use and the method for controlling fungi, insects/acari and weeds of the compounds of the present invention.

IPC Classes  ?

• C07D 417/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles

Abstract

Disclosed are an N-(aryl alkyl) aryloxy phenoxy carboxylic acid amide compound expressed by formula (I) and a preparation method and application thereof. Ar1, Ar2, R1, R2, R3, and n in formula (I) are defined as given in the specification. The compound of formula (I) according to the present invention has weeding and/or sterilizing, insecticidal, and acaricidal bioactivities. Some compounds have a very high herbicidal activity, and desirable effects can be achieved with a dosage of 15 to 75 g effective components per hectare.

IPC Classes  ?

• C07D 417/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 277/32 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
• C07D 213/643 - 2-PhenoxypyridinesDerivatives thereof
• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 413/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 43/60 - 1,4-DiazinesHydrogenated 1,4-diazines
• A01N 43/76 - 1,3-OxazolesHydrogenated 1,3-oxazoles
• A01P 13/00 - HerbicidesAlgicides
• A01P 3/00 - Fungicides
• A01P 7/04 - Insecticides
• A01P 7/02 - Acaricides

Abstract

Disclosed in the present invention is a N-pyridine(hetero)aromatic amide compound of formula (I) and a preparation method and use thereof In the formula, Ar, R1, R2, R3, m and X have definitions as given in the description. The compound of formula (I) of the present invention has fungicidal and/or phytocidal, insecticidal and acaricidal bioactivities.

IPC Classes  ?

• C07D 213/75 - Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
• C07D 213/76 - Nitrogen atoms to which a second hetero atom is attached
• C07D 417/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 417/14 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing three or more hetero rings
• C07D 213/82 - AmidesImides in position 3
• C07D 401/12 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
• C07D 401/14 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• A01N 43/828 - 1,2,3-Oxa(thia)diazolesHydrogenated 1,2,3-oxa(thia)diazoles
• A01N 43/56 - 1,2-DiazolesHydrogenated 1,2-diazoles
• A01P 3/00 - Fungicides
• A01P 7/04 - Insecticides
• A01P 7/02 - Acaricides
• A01P 13/00 - HerbicidesAlgicides

Abstract

Disclosed are a N-pyridine amide compound shown in formula (I), a preparation method therefor, and an application thereof. In formula (I), R, R1, R2, R3, and m all have the definitions given in the specification. The compound shown in formula (I) of the present invention has the biological activity of sterilization and/or pest killing, mite killing, and weeding.

IPC Classes  ?

• C07D 213/75 - Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
• A01N 43/40 - Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
• A01P 3/00 - Fungicides
• A01P 7/02 - Acaricides
• A01P 7/04 - Insecticides
• A01P 13/00 - HerbicidesAlgicides

Abstract

Disclosed are thiazole methylamino pyridine compounds as shown by formula (I) having fungicidal, insecticidal/acaricidal, and phytocidal bioactivity, the preparation method thereof, the fungicidal, insecticidal/acaricidal, and herbicide compositions containing the compounds, and the use and the method for controlling fungi, insects/acari and weeds using the compounds.

IPC Classes  ?

• C07D 417/12 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
• A01N 43/78 - 1,3-ThiazolesHydrogenated 1,3-thiazoles
• A01P 3/00 - Fungicides
• A01P 7/04 - Insecticides
• A01P 7/02 - Acaricides
• A01P 13/00 - HerbicidesAlgicides