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2025
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Invention
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Methods of manufacturing a bifunctional compound. This disclosure pertains to the preparation of ... |
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Invention
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Pharmaceutical formulations of an androgen receptor-targeting protein degrader. The present discl... |
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Invention
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Pharmaceutical formulations of an androgen receptor-targeting protein degrader.
The present disc... |
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Invention
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Crystalline forms of a compound for the targeted degradation of bcl6. The present disclosure rela... |
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Invention
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Benzimidazole and benzimidazolone based protac compounds for the targeted degradation of leucine ... |
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Invention
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Methods of manufacturing a bifunctional compound.
This disclosure pertains to the preparation of... |
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Invention
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Methods of manufacturing an androgen receptor protein degrader.
This disclosure pertains to meth... |
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Invention
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Methods of manufacturing an androgen receptor protein degrader. This disclosure pertains to metho... |
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G/S
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Pharmaceutical preparations for the treatment of cancer. |
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G/S
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Pharmaceutical preparations for the treatment of cancer |
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Invention
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Cereblon ligands and bifunctional compounds comprising the same.
The description relates to cere... |
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Invention
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Modulators of bcl6 proteolysis and associated methods of use. This application pertains to the us... |
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2024
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Invention
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Rapidly accelerating fibrosarcoma protein degrading compounds and associated methods of use.
Bif... |
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Invention
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Methods of treating breast cancer with tetrahydronaphthalene derivatives as estrogen receptor deg... |
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Invention
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Compounds and methods for the targeted degradation of androgen receptor.
The present disclosure ... |
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Invention
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Synthesis of leucine-rich repeat kinase 2 modulators. Provided are methods for synthesizing compo... |
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Invention
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Use of androgen receptor degrader for the treatment of spinal and bulbar muscular atrophy.
This ... |
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Invention
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Use of androgen receptor degrader for the treatment of spinal and bulbar muscular atrophy. This d... |
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Invention
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Rapidly accelerated fibrosarcoma (raf) degrading compounds and associated methods of use.
Provid... |
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G/S
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Pharmaceutical preparations for the treatment of cancer. |
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Invention
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Compounds and methods for the targeted degradation of bromodomain-containing proteins.
The prese... |
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Invention
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Crystalline and amorphous forms of a compound for the targeted degradation of estrogen receptor. ... |
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G/S
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Pharmaceutical preparations for the treatment of cancer Medical informational services, including... |
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Invention
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Tetrahydronaphthalene and tetrahydroisoquinoline derivatives as estrogen receptor degraders.
The... |
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Invention
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Vepdegestrant dosage regimen in cyp3a-inducer treatment in cancer. The invention relates to a met... |
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Invention
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Indazole based compounds and associated methods of use.
Bifunctional compounds, which find utili... |
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Invention
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Dgk targeting compounds and uses thereof. e.ge.g., cancer) and viral infections. |
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Invention
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Hpk1 targeting compounds and uses thereof. Described herein are compounds that modulate hematopoi... |
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Invention
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Compounds useful in the treatment of kras mediated disorders. e.g.e.g., compounds of Formula (I))... |
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Invention
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Compounds and methods for the targeted degradation of androgen receptor.
This disclosure pertain... |
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Invention
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Compounds and methods for the targeted degradation of androgen receptor. This disclosure pertains... |
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G/S
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Pharmaceutical preparations for the treatment of cancer |
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Invention
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Combinations of estrogen receptor degraders and cdk7 inhibitors for the treatment of cancer. Disc... |
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Invention
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Methods of manufacturing a bifunctional compound, ultrapure forms of the bifunctional compound, a... |
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Invention
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Solid oral dosage forms of estrogen receptor degraders. Disclosed herein are solid oral dosage fo... |
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Invention
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Combinations of estrogen receptor degraders and akt inhibitors. Disclosed herein are methods for ... |
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Invention
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Bavdegalutamide for treating prostate cancer without ar l702h mutation. This disclosure pertains ... |
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Invention
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Use of an androgen receptor degrader protac for the treatment of prostate cancer. The present app... |
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Invention
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Egfr proteolysis targeting chimeric molecules and associated methods of use.
The present inventi... |
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Invention
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Crystalline forms of a compound for the targeted degradation of the androgen receptor.
The prese... |
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Invention
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Crystalline forms of a compound for the targeted degradation of the androgen receptor. The presen... |
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Invention
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Dosage regimens of estrogen receptor degraders. Disclosed herein are methods for treating cancer ... |
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Invention
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Modulators of bcl6 proteolysis and associated methods of use.
Bifunctional compounds, which find... |
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Invention
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Dosage regimens of estrogen receptor degraders in combination with an mtor inhibitor. Disclosed h... |
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Invention
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Cereblon-based kras degrading protacs and uses related thereto. Provided herein are compounds tha... |
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Invention
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Modulators of bcl6 proteolysis and associated methods of use.
This application pertains to the u... |
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2023
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Invention
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Imide-based modulators of proteolysis and associated methods of use.
The description relates to ... |
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Invention
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Bavdegalutamide and combinations thereof for use in treating prostate cancer.
This disclosure pe... |
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Invention
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Compounds and methods for the targeted degradation of kras.
Bifunctional compounds, which find u... |
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2022
|
Invention
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Brm targeting compounds and associated methods of use.
The present disclosure relates to bifunct... |
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Invention
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Brm degrading compounds and associated methods of use.
The present disclosure relates to bifunct... |
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G/S
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Pharmaceutical preparations for use in treating oncology, immunology, and central nervous system ... |
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G/S
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Pharmaceutical preparations for use in treating oncology,
immunology, and inflammatory diseases,... |
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2021
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G/S
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Agricultural products development |
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G/S
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Bi-functional small molecules that mediate targeted protein degradation through the ubiquitin pro... |
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G/S
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Pharmaceutical preparations for use in treating oncology, immunology, and inflammatory diseases, ... |
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2020
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G/S
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Pharmaceutical products development of new small molecules aimed at degrading disease-causing cel... |
