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2016
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Invention
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Furo[3, 2-b] pyrr0l-3-ones as cathespin s inhibitors.
A first aspect of the invention relates to... |
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2015
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Invention
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Furo [3, 2-b] pyrr0l-3-0nes as cathespin s inhibitors.
A first aspect of the invention relates t... |
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Invention
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Piperazine compounds.
A compound of formula (I), or a pharmaceutically acceptable salt, hydrate,... |
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2013
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Invention
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Furo[3, 2-b] pyrrol-3-ones as cathespin s inhibitors. A first aspect of the invention relates to ... |
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2010
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Invention
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Piperazine compounds. A compound of formula (I), or a pharmaceutically acceptable salt, hydrate, ... |
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Invention
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Furo[3. 2-b] pyrrol derivatives. 3-8 cycloalkyl. The invention further relates to pharmaceutical ... |
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2009
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Invention
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Tetrahydrofuro [3, 2-b] pyrrol-3-one derivatives as inhibitors of cysteine proteases. A compound ... |
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Invention
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Furo [3, 2-b] pyrr0l-3-0nes as cathepsin s inhibitors. A first aspect of the invention relates to... |
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Invention
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Compounds. A first aspect of the invention relates to a compound of formula (I), or a pharmaceuti... |
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Invention
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Furo[3,2-b]pyrrol-3-one derivatives and their use as cysteinyl proteinase inhibitors. The present... |
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Invention
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Tetrahydrofuro[3,2-b] pyrrol-3-ones as cathepsin k inhibitors. The present invention relates to c... |
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Invention
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Furo[3,2-b] pyrrol-3-one derivatives and their use as cysteinyl proteinase inhibitors. 3-8 cycloa... |
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Invention
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Furo[3, 2-b] pyrrol derivatives. 3-8 cycloalkyl. The invention further relates to pharmaceutical ... |
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Invention
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Tetrahydrofuro(3,2-b) pyrrol-3-one derivatives as inhibitors of cysteine proteinases. A compound ... |
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Invention
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Tetrahydrofuro (3, 2 -b) pyrrol- 3 -one derivatives as inhibitors of cysteine proteinases. A comp... |
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2008
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Invention
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Inhibitors of cruzipain and other cysteine proteases.
Compounds of general formula (I) or genera... |
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Invention
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Preparation of diazapentalene derivatives via epoxydation of dihydropyrroles.
The present invent... |
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2007
|
Invention
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Furo [3, 2-b] pyrrol derivatives. The present invention relates to compounds of formula (I), and ... |
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Invention
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Tetrahydrofuro [3, 2-b] pyrr0l-3-ones as cathepsin k inhibitors. The present invention relates to... |
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|
Invention
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Tetrahydrofuro [3, 2 -b] pyrr0l-3-ones as cathepsin k inhibitors. The present invention relates t... |
|
|
Invention
|
Furo [3,2-b] pyrrol-3-one derivatives and their use as cysteinyl proteinase inhibitors. The prese... |
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|
Invention
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Tetrahydrofuro (3, 2-b) pyrrol-3-one derivatives as inhibitors of cysteine proteinases. Compounds... |
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Invention
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Tetrahydrofuro [3, 2-b] pyrr0l-3-0ne intermediates. The present invention relates to a process fo... |
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2006
|
Invention
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Biologically active compounds. The present invention relates to compounds of formula (I), and pha... |
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Invention
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Preparation of diazapentalene derivatives via epoxydation of dihydropyrroles. The present inventi... |
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Invention
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Method of producing conjugate vaccines. The present invention relates to a method of production o... |
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2004
|
Invention
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Cyclic 2-carbonylaminoketones as inhibitors of cruzipain and other cysteine proteases. Compounds ... |
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Invention
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Inhibitors of cruzipain and other cysteine proteases. Compounds of general formula (I):
m, Z and... |
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Invention
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Inhibitors of cruzipain and other cysteine proteases. m, Z and U are as defined in the specificat... |
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2003
|
Invention
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Biologically active compounds.
Compounds of general formula (I)
wherein Z=CR3R4, where R3... |
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Invention
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Biologically active compounds. Compounds of general formula (I) wherein: Z = CR3R4, where R3 and ... |
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Invention
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Charge-balanced chemoselective linkers.
Compounds according to general formulae (Ia to Ie) where... |
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Invention
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Charge-balanced chemoselective linkers. Compounds according to general formulae (Ia to Ie) wherei... |
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Invention
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Enzyme substrates for the determination of activity of staphylococcus sp. extracellular protease.... |
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Invention
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Fmdv leader peptidase assay. Footᇁandᇁmouth disease virus ࿈FMDV) leader peptidase activity i... |
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Invention
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Assay for staphylococcus sp. extracellular cysteine peptidase activity. Staphylococcus sp. extrac... |
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2002
|
Invention
|
Inhibitors of cruzipain and other cysteine proteases. Compounds of general formula (I) or general... |
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Invention
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Inhibitors of cruzipain and other cysteine proteases. Compounds of general formula (I): wherein R... |
